Regioselective C 2 sulfonylation of indoles mediated by molecular iodine

Praewpan Katrun; Charoensak Mueangkaew; Manat Pohmakotr; Vichai Reutrakul; Thaworn Jaipetch; Darunee Soorukram; Chutima Kuhakarn

doi:10.1021/jo402831k

Regioselective C 2 sulfonylation of indoles mediated by molecular iodine

Praewpan Katrun
, Charoensak Mueangkaew
, Manat Pohmakotr
, Vichai Reutrakul
, Thaworn Jaipetch
, Darunee Soorukram
, Chutima Kuhakarn

Mahidol University
Mahidol University

Research output: Contribution to journal › Article › peer-review

119 Citations (Scopus)

Abstract

A facile and general method for regioselective C2 sulfonylation reaction of indoles mediated by iodine is described. The 2-sulfonylated products were obtained up to 96% yield under mild reaction conditions (room temperature, 2 h).

Original language	English
Pages (from-to)	1778-1785
Number of pages	8
Journal	Journal of Organic Chemistry
Volume	79
Issue number	4
DOIs	https://doi.org/10.1021/jo402831k
Publication status	Published - 21 Feb 2014
Externally published	Yes

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@article{c82a2c79597f491f8e08b8462ed5c4e3,

title = "Regioselective C 2 sulfonylation of indoles mediated by molecular iodine",

abstract = "A facile and general method for regioselective C2 sulfonylation reaction of indoles mediated by iodine is described. The 2-sulfonylated products were obtained up to 96\% yield under mild reaction conditions (room temperature, 2 h).",

author = "Praewpan Katrun and Charoensak Mueangkaew and Manat Pohmakotr and Vichai Reutrakul and Thaworn Jaipetch and Darunee Soorukram and Chutima Kuhakarn",

year = "2014",

month = feb,

day = "21",

doi = "10.1021/jo402831k",

language = "English",

volume = "79",

pages = "1778--1785",

journal = "Journal of Organic Chemistry",

issn = "0022-3263",

publisher = "American Chemical Society",

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T1 - Regioselective C 2 sulfonylation of indoles mediated by molecular iodine

AU - Katrun, Praewpan

AU - Mueangkaew, Charoensak

AU - Pohmakotr, Manat

AU - Reutrakul, Vichai

AU - Jaipetch, Thaworn

AU - Soorukram, Darunee

AU - Kuhakarn, Chutima

PY - 2014/2/21

Y1 - 2014/2/21

N2 - A facile and general method for regioselective C2 sulfonylation reaction of indoles mediated by iodine is described. The 2-sulfonylated products were obtained up to 96% yield under mild reaction conditions (room temperature, 2 h).

AB - A facile and general method for regioselective C2 sulfonylation reaction of indoles mediated by iodine is described. The 2-sulfonylated products were obtained up to 96% yield under mild reaction conditions (room temperature, 2 h).

UR - https://www.scopus.com/pages/publications/84894576414

U2 - 10.1021/jo402831k

DO - 10.1021/jo402831k

M3 - Article

C2 - 24475946

AN - SCOPUS:84894576414

SN - 0022-3263

VL - 79

SP - 1778

EP - 1785

JO - Journal of Organic Chemistry

JF - Journal of Organic Chemistry

IS - 4

ER -

Regioselective C 2 sulfonylation of indoles mediated by molecular iodine

Abstract

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